Recent TYDOCK PHARMA Publications

2014

D. Farina, F. Spyrakis, A. Venturelli, S. Cross, D. Tondi, M.P. Costi: "The inhibition of estende spectrum b-lactamases: hits and leads." Curr. Med. Chem., 2014, 21, 1405-34.

Pellati Federica, Mascolo Danilo, Venturelli Alberto, Barbato Amedeo, Davide Righi, Paco Castaldi “ Nuovo Trattamento assistito da Microonde per la produzione di miscele arricchite di policosanoli da matrici cerose”  Patent MI 201400030, 27 Febbraio 2014.

Marco Consales, Giuseppe Quero, Simona Zuppolini, Lucia Sansone, Anna Borriello, Michele Giordano, Alberto Venturelli, Andrea Cusano “Reflection -type long period grating biosensor for the detection of drug resistant bacteria: The Opto-bacteria project” PROCEEDINGS OF SPIE VOLUME 9157 Volume Number: 9157, Softcover: 390 papers (1742) pages, ISBN: 9781628411751, 22 May 2014.

Tondi D #, Venturelli A #, Bonnet R, Pozzi C, Shoichet BK, Costi MP: “Targeting class A and C serine β-lactamases with a broad-spectrum boronic acid derivative” J Med Chem. 2014 Jun 26;57(12):5449-58 # These authors contributed equally.

F. Spyrakis, S. Cross, G. Cruciani, M. Santucci, D. Farina, A. Venturelli, M.P. Costi. “New ligands for detecting drug resistant bacteria” in 20th EuroQSAR, Understanding Chemical-Biological Interactions, St-Petersburg, Russia, August 31-September 4, 2014. Poster session.

9th June 2014 – 11th June 2014: 8th Annual Meeting "New Perspectives in Medicinal Chemistry” NPCF8: Matteo Santucci, A. Venturelli, F. Spyrakis, D. Farina, A. Cusano, A. Borriello, S. Zuppolini, L. Sansone, M.P. Costi; “Ligands Discovery: Molecular Tool for Beta-Lactamases detection in biological matrix”, Parma, Italy.

18th December 2014: Italian Chemical Society-Emilia Romagna Section: XV Meeting of Emilia Romagna Chemistry: Matteo Santucci, Francesca Spyrakis, Nageswara Rao Nalajala, Alberto Venturelli, Simon Cross, Jesus Blazquez, Anna Borriello, Simona Zuppolini, Maria Paola Costi; “New ligands for beta-lactamases biosensing”; Parma; Italy.

 

2015/2016

Neres J, Hartkoorn RC, Chiarelli LR, Gadupudi R, Pasca MR, Mori G, Venturelli A, Savina S, Makarov V, Kolly GS, Molteni E, Binda C, Dhar N, Ferrari S, Brodin P, Delorme V, Landry V, de Jesus Lopes Ribeiro AL, Farina D, Saxena P, Pojer F, Carta A, Luciani R, Porta A, Zanoni G, De Rossi E, Costi MP, Riccardi G, Cole ST: “2-carboxyquinoxalines kill mycobacterium tuberculosis through noncovalent inhibition of DprE1”. ACS Chem Biol. 2015 Mar 20;10(3):705-14. doi: 10.1021/cb5007163. Epub 2014 Dec 9.

D. Tondi, S. Cross, A. Venturelli, M.P. Costi, G. Cruciani, F. Spyrakis: “Decoding the structural basis for carbapenem hydrolysis by class A beta-lactamases: fishing for a pharmacophore.” Curr Drug Targets. 2015 Sep 30. [Epub ahead of print]

Quero, Giuseppe; Zuppolini, Simona; Consales, Marco; Diodato, Laura; Vaiano, Patrizio; Venturelli, Alberto; Santucci, Metteo; Spyrakis, Francesca; Costi, Maria Paola; Giordano, Michele; Borriello, Anna; Cutolo, Antonello; Cusano, Andrea.. "Long Period Fiber Grating Working in Reflection Mode as Valuable Biosensing Platform for the Detection of Drug Resistant Bacteria".  Sensor and Actuators B Chemical 230, February 2016.

Antonio Quotadamo, Pasquale Linciano, Paolo Davoli, Donatella Tondi, Maria Paola Costi *, Alberto Venturelli1*An Improved Synthesis of CENTA, Chromogenic Substrate for β-Lactamases. Synlett Accepted. 2016

 

 

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