Recent TYDOCK PHARMA Publications

Neres J, Hartkoorn RC, Chiarelli LR, Gadupudi R, Pasca MR, Mori G, Venturelli A, Savina S, Makarov V, Kolly GS, Molteni E, Binda C, Dhar N, Ferrari S, Brodin P, Delorme V, Landry V, de Jesus Lopes Ribeiro AL, Farina D, Saxena P, Pojer F, Carta A, Luciani R, Porta A, Zanoni G, De Rossi E, Costi MP, Riccardi G, Cole ST. “2-carboxyquinoxalines kill mycobacterium tuberculosis through noncovalent inhibition of DprE1”. ACS Chem Biol. 2015 Mar 20;10(3):705-14.

Maxwell A: F1000Prime Recommendation of Evaluation [Neres J et al., ACS Chem Biol 2014]. In F1000Prime, 09 Jan 2015; DOI: 10.3410/f.725248139.793502885.

G. Quero, M. Consales, P.Vaiano, A. Cusano, M. Giordano,  S. Zuppolini, L. Diodato, A. Borriello, A. Venturelli, M.P. Costi. “Reflection-type long period grating biosensor for the detection of drug resistant bacteria: The Opto-bacteria Project”. AISEM Annual Conference, 2015 XVIII, IEEE Conference Publications.

D. Tondi, S. Cross, A. Venturelli, M.P. Costi, G. Cruciani, F. Spyrakis. “Decoding the structural basis for carbapenem hydrolysis by class A beta-lactamases: fishing for a pharmacophore.” Curr Drug Targets. 2016;17(9):983-1005.

Quero, Giuseppe; Zuppolini, Simona; Consales, Marco; Diodato, Laura; Vaiano, Patrizio; Venturelli, Alberto; Santucci, Metteo; Spyrakis, Francesca; Costi, Maria Paola; Giordano, Michele; Borriello, Anna; Cutolo, Antonello; Cusano, Andrea."Long Period Fiber Grating Working in Reflection Mode as Valuable Biosensing Platform for the Detection of Drug Resistant Bacteria". Sensor and Actuators B Chemical 230, February 2016.

Antonio Quotadamo, Pasquale Linciano, Paolo Davoli, Donatella Tondi, Maria Paola Costi, Alberto Venturelli. “An Improved Synthesis of CENTA, Chromogenic Substrate for β-Lactamases”. Synlett 2016; 27(17): 2447-2450 DOI: 10.1055/s-0035-1562454.

Luciani, Rosaria; Saxena, Puneet; Surade, Sachin; Santucci, Matteo; Venturelli, Alberto; Borsari, Chiara; Marverti, Gaetano; Ponterini, Glauco; Ferrari, Stefania; Blundell, Tom L.; Costi, Maria Paola. “Virtual screening and X-ray crystallography Identify non-substrate analog inhibitors of Flavin-dependent Thymidylate Synthase”. J. Med. Chem. 2016, 59, 19, 9269-9275.

Chiara Borsari, Stefania Ferrari, Alberto Venturelli, Maria Paola Costi “Target-based approaches for the discovery of new antimycobacterial drugs”. Drug Discov Today 2017 Mar;22(3):576-584.

Simona Zuppolini, Giuseppe Quero, Marco Consales, Laura Diodato, Patrizio Vaiano, Alberto Venturelli, Matteo Santucci, Francesca Spyrakis, Maria P. Costi, Michele Giordano, Antonello Cutolo, Andrea Cusano, and Anna Borriello. “Label-free fiber optic optrode for the detection of class C β-lactamases expressed by drug resistant bacteria”. Biomedical Optics Express Vol. 8, Issue 11, pp. 5191-5205 (2017).

Panecka-Hofman J, Pöhner I, Spyrakis F, Zeppelin T, Di Pisa F, Dello Iacono L, Bonucci A, Quotadamo A, Venturelli A, Mangani S, Costi MP, Wade RC. “Comparative mapping of on-targets and off-targets for the discovery of anti-trypanosomatid folate pathway inhibitors”. Biochim Biophys Acta Gen Subj. 2017 Dec;1861(12):3215-3230.

Luca Ferrari , Luigi Rovati , Maria Paola Costi , Alberto Venturelli , Rosaria Luciani , and Stefano CattiniOn the feasibility of a CENTA-based biosensor to measure antibiotics concentration in milk”. Optics InfoBase Conference Papers (2017) Part F61-ECBO 2017

L Ferrari, L Rovati, MP Costi, R Luciani, A Venturelli, S Cattini "Feasibility Study on a Measurement Method and a Portable Measuring System to Estimate the Concentration of Cloxacillin and β-Lactamase in Milk".  Journal of Sensors Vol. 2017, Article ID 5742359, 11 pages, 2017. doi:10.1155/2017/5742359.

Matteo Santucci, Francesca Spyrakis, Simon Cross, Antonio Quotadamo, Davide Farina, Donatella Tondi, Jean-Denis Docquier, Filomena Croce, Ana Isabel Prieto, Claudia Ibacache, Jesús Blázquez , Alberto Venturelli*, Gabriele Cruciani,* Maria Paola Costi*.  “Computational and biological profile of boronic acids for the detection of cellular serine- and metallo-b-lactamases”. Scientific Report 7 (1), 17716, 2017.

Maria Paola Costi, Matteo Santucci, Francesca Spyrakis, Simon Cross, Davide Farina, Donatella Tondi, Antonio Quotadamo, Jean-Denis Docquier, Filomena Croce, Ana Isabel Prieto, Claudia Ibacache, Jesús Blázquez, Alberto Venturelli, Gabriele Cruciani. pag.217-218. Organization of the Book of Abstracts: Ana Laço, José Luis Capelo, Carlos Lodeiro “Proceeding of the 2nd IC2AR Conference on Antibiotic resistance. O 03C - Multiligand approach to the identification of resistant strains overexpressing beta-lactamase”. ISBN: 978-989-99639-3-1. Printed by Proteomass (Portugal) Printage: 50 copies (paper) Caparica, Portugal, 2017.

Chiara Borsari, Antonio Quotadamo, StefaniaFerrari, AlbertoVenturelli, AnabelaCordeiro-da-           Silva, Nuno Santarem, Maria PaolaCosti. “Chapter Two - Scaffolds and Biological Targets Avenue to Fight Against Drug Resistance in Leishmaniasis.” Annual Reports in Medicinal Chemistry Volume 51, 2018, Pages 39-95.

Francesca Spyrakis, Donatella Tondi, Giuseppe Celenza, Giulia D’Arrigo, Eleonora Gianquinto, Matteo Santucci, Simon Cross, Pierangelo Bellio, Laura Cendron, Jean-Denis Docquier, Jesùs Blàzquez, Alberto Venturelli, Gabriele Cruciani, Maria Paola Costi. “In silico/in vitro approaches for the identification of new carbapenemase inhibitors”   Poster Ref. Chem. Lett Vol. 9, 45-50, 2018.

Moraes CB, Witt G, Kuzikov M, Ellinger B, Calogeropoulou T, Prousis KC, Mangani S, Di Pisa F, Landi G, Iacono LD, Pozzi C, Freitas-Junior LH, Dos Santos Pascoalino B, Bertolacini CP, Behrens B, Keminer O, Leu J, Wolf M, Reinshagen J, Cordeiro-da-Silva A, Santarem N, Venturelli A, Wrigley S, Karunakaran D, Kebede B, Pöhner I, Müller W, Panecka-Hofman J, Wade RC, Fenske M, Clos J, Alunda JM, Corral MJ, Uliassi E, Bolognesi ML, Linciano P, Quotadamo A, Ferrari S, Santucci M, Borsari C, Costi MP, Gul S.   “Accelerating Drug Discovery Efforts for Trypanosomatidic Infections Using an Integrated Transnational Academic Drug Discovery Platform”  SLAS Discov. 2019 Mar;24(3):346-361.

Laura Cendron, Antonio Quotadamo, Lorenzo Maso, Pierangelo Bellio, Martina Montanari, Giuseppe Celenza, Alberto Venturelli, Maria Paola Costi, and Donatella Tondi. “X-ray-crystallography deciphers the activity of broad spectrum boronic acid -Lacatamases inhibitors”. ACS Med. Chem. Lett., 2019, 10 (4), pp 650–655 Publication Date (Web): March 27, 2019 (Letter).

Alberto Venturelli, Virginia Brighenti, Danilo Mascolo, Federica Pellati. “A new strategy based on microwave-assisted technology for the extraction and purification of beeswax policosanols for pharmaceutical purposes and beyond” J Pharm Biomed Anal. 2019 Aug 5;172:200-205.

Antonio Quotadamo, Pasquale Linciano, Maria Paola Costi, Alberto Venturelli*. “Optimization of N-alkylation in the synthesis of methotrexate and pteridine-based derivatives under microwave-irradiation”.  Chemistry Select 4(15):4429 · April 2019.

 

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